85-2076-95　SR95531 (Gabazine, GABAA Receptor Antagonist, SR-95531, Gabazine, SR95531, SR 95531) 10mg　CAS No:104104-50-9　217808

特徴

• A selective, competitive antagonist of GABAA receptor (IC50 = 440nM) that does not affect pentobarbitone or etomidate- induced currents even at high concentrations (~100uM). Also shown to block glycine receptors, but with low affinity (Kb = 190uM).
• Synonyms:GABAA Receptor Antagonist, SR-95531, Gabazine, SR95531, SR 95531
• Primary Target:GABA-A
• Primary Target IC50:440nM
• Solubility:Water (25mM)
• Proton NMR:Conforms to structure
• Elemental Analysis:C% :47.50-50.50%H%: 4.00-6.00%N%: 10.00-13.00%
• Water Molecules:≤1.0mol
• Appearance:Supplied as a white solid.
• Purity:≥98% (HPLC)
• Storage and Stability:Lyophilized powder may be stored at 4°C. Do not freeze. Stable for 6 months after receipt at 4°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap.