A very potent and selective delta opioid receptor agonist (IC50 = 0.32uM). Shown to induce dose- and time-dependent antinociception after i.c.v., i.th. and i.p. administration in mice. Widely used in studies of depression and inflammatory injuries. It is also reported to be acted upon heteromeric u-d receptors.
Synonyms:δ Opioid Receptor Agonist, SNC80
Molecular Formula:C₂₈H₃₉N₃O₂
Solubility:DMSO or 1N HCl
Primary Target:Delta opioid receptor
Primary Target IC50:0.32u
Purity:≥98% (HPLC)
Form:Supplied as a cream solid.
Storage and Stability:May be stored at 4°C for short-term only. Long-term storage is recommended at -20°C. Stable for 1 year after receipt. Protect from light. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
