A highly potent antagonist slightly selective for NR2A over other subtype nMDA receptors (Ki = 0.041, 0.27, 0.63 and 1.99uM for nMDA subtypes NR2A, NR2B, NR2C, and NR2D, respectively). Commonly used for various research in brain functions and disorders that neurotransmissions via nMDA receptors are involved.
Primary Target Ki:0.041, 0.27, 0.63 and 1.99 →M for NMDA subtypes NR2A, NR2B, NR2C, and NR2D, respectively.
Purity:≥98% (NMR)
Form:Supplied as an off-white solid.
Storage and Stability:May be stored at 4°C. For long-term storage, aliquot and store at 4°C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.