Selective dopamine D3 receptor agonist (Ki = 2.3nM) with an 18-fold selectivity over long dopamine receptors (D2L) and exhibited only weak affinity for D4.2 receptors (Ki = 169nM). Commonly used to reproduce cocaine's discriminative stimulus effects and also in peripheral systemic studies of hypertension.
Molecular Formula:C₁₄H₁₉NO₃•HCl
Solubility:H2O
Primary Target:D3
Primary Target Ki:2.3nM
Storage and Stability:Store at -20°C under inert atmosphere. For maximum recovery of product, centrifuge the original vial prior to removing the cap.
