85-2072-25　CPCCOEt ((E)-Ethyl 1,1a,7,7a-tetrahydro-7-(hydroxyimino)cyclopropa[b]chromene-1a-carboxylate, mGlu1 Antagonist, CPCCOEt) 5mg　CAS No:179067-99-3　217283

特徴

• A potent, negative allosteric modulator selective for mGlu1 receptors (IC50 = 6.5uM). No effect on other mGlu subtype receptors and ionotropic glutamate receptors at concentrations less than 100uM. Acts by inhibiting an intramolecular interaction between the agonist-bound extracellular domain and the transmembrane domain. Widely used for studies related to peripheral pain and central pain pathways.
• Formula:C13H13NO4
• Solubility:DMSO
• Primary Target:mGlu1 receptors
• Molar Mass:247.25
• Storage and Stability:May be stored at 4°C. For long-term storage, aliquot and store at 4°C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.

仕様

• Size：5mg
• Grade：Highly Purified
• Purity：~98% (HPLC)
• Form：Supplied as a white powder.
• Molecular Formula：C13H13NO4
• Molecular Weight Non Ab：247.25
• EU Commodity Code：38220090
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• 製品の仕様は予告なく変更になる場合がございます。最新仕様はメーカーホームページをご確認ください。
• CAS No ：179067-99-3

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