Protein kinase D (PKD) inhibitor (IC50 values are 0.6, 0.7 and 3.2um for PKD2, PKD3 and PKD1 respectively). Cell permeable (EC50=10um for PKD1 inhibition). ATP-competitive.
Formula:C22H21ClN2O3
Solubility:DMSO (~50mM)
Molecular Weight:~396.87
Storage and Stability:Store at RT. Stable for 12 months.