Highly selective ETB-receptor antagonist (IC50=1.2nM). BQ 788 is an endothelin type B (ETB) receptor antagonist and is a potential antidote for the cardiovascular toxicity with hypotension and bradycardia.
Appearance:White Solid
Purity:~90%
Melting Point:>144°C (dec.)
Storage:4°C
Solubility:DMSO (Slightly)
Storage and Stability:Powder may be stored at 4°C for short-term only. Stable for 12 months at -20°C. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.
